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GLP-1R Agonist DMB
CAS No. 281209-71-0
GLP-1R Agonist DMB( —— )
Catalog No. M34861 CAS No. 281209-71-0
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 104 | In Stock |
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| 5MG | 133 | In Stock |
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| 10MG | 203 | In Stock |
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| 25MG | 323 | In Stock |
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| 50MG | 531 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGLP-1R Agonist DMB
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NoteResearch use only, not for human use.
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Brief DescriptionGLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
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DescriptionGLP-1R agonist 2 (compound 2) is a potent GLP-1R agonist. GLP-1R agonist 2 has the potential for the research of metabolic diseases like Type2 Diabetes and Obesity.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetGlucagon Receptor
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RecptorGlucagon Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number281209-71-0
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Formula Weight348.25
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Molecular FormulaC13H15Cl2N3O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (71.79 mM; Ultrasonic (<60°C)
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SMILESCC(C)(C)Nc1nc2cc(Cl)c(Cl)cc2nc1S(C)(=O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Girdhar K, et al. Novel insights into the dynamics behavior of glucagon-like peptide-1 receptor with its small molecule agonists. J Biomol Struct Dyn. 2019 Sep;37(15):3976-3986.?
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