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N-desmethyl Olanzapine
CAS No. 161696-76-0
N-desmethyl Olanzapine( —— )
Catalog No. M34784 CAS No. 161696-76-0
N-desmethyl Olanzapine is a metabolite of the atypical antipsychotic compound Olanzapinec, which is formed through the oxidative metabolism of olanzapine by the cytochrome 450 (CYP) isoenzyme CYP1A2.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 164 | In Stock |
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| 10MG | 238 | In Stock |
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| 25MG | 506 | In Stock |
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| 50MG | 715 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameN-desmethyl Olanzapine
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NoteResearch use only, not for human use.
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Brief DescriptionN-desmethyl Olanzapine is a metabolite of the atypical antipsychotic compound Olanzapinec, which is formed through the oxidative metabolism of olanzapine by the cytochrome 450 (CYP) isoenzyme CYP1A2.
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DescriptionN-Desmethylolanzapine is an antipsychotic drug.The formation of N-Desmethylolanzapine correlates with the level and activityof human liver flavin-containing monooxygenase (FMO3). N-Desmethylolanzapinecan be used in the study of antipsychotic drugs .
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetP450
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RecptorP450 | Drug Metabolite
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Research Area——
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Indication——
Chemical Information
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CAS Number161696-76-0
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Formula Weight298.41
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Molecular FormulaC16H18N4S
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Purity>98% (HPLC)
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Solubility——
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SMILESCc1cc2c(Nc3ccccc3N=C2N2CCNCC2)s1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ring BJ, et al. Identification of the human cytochromes P450 responsible for the in vitro formation of the major oxidative metabolites of the antipsychotic agent olanzapine. J Pharmacol Exp Ther. 1996 Feb;276(2):658-66.?
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