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LY2033298
CAS No. 886047-13-8
LY2033298( —— )
Catalog No. M34325 CAS No. 886047-13-8
LY2033298, a positive allosteric modulator of muscarine M4 receptor, enhances the inhibitory effect of oximoline on light-induced phase shift in circadian activity in hamsters and can be used in neurosystem-related diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 204 | In Stock |
|
| 10MG | 347 | In Stock |
|
| 25MG | 562 | In Stock |
|
| 50MG | 797 | In Stock |
|
| 100MG | 1070 | In Stock |
|
| 200MG | 1442 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLY2033298
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NoteResearch use only, not for human use.
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Brief DescriptionLY2033298, a positive allosteric modulator of muscarine M4 receptor, enhances the inhibitory effect of oximoline on light-induced phase shift in circadian activity in hamsters and can be used in neurosystem-related diseases.
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DescriptionLY 2033298 is a selective positive allosteric modulator of the muscarinic M4 receptor. LY 2033298 can be used in the study of psychiatric disorders.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetAChR
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RecptorAChR
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Research Area——
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Indication——
Chemical Information
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CAS Number886047-13-8
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Formula Weight311.79
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Molecular FormulaC13H14ClN3O2S
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Purity>98% (HPLC)
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Solubility——
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SMILESCOc1nc2sc(C(=O)NC3CC3)c(N)c2c(C)c1Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chan WY, et al. Allosteric modulation of the muscarinic M4 receptor as an approach to treating schizophrenia. Proc Natl Acad Sci U S A. 2008 Aug 5;105(31):10978-83.?
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