IK-862

CAS No. 478911-60-3

IK-862( —— )

Catalog No. M34281 CAS No. 478911-60-3

IK-862 is a selective inhibitor of TACE (ADAM17).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 848 In Stock
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Biological Information

  • Product Name
    IK-862
  • Note
    Research use only, not for human use.
  • Brief Description
    IK-862 is a selective inhibitor of TACE (ADAM17).
  • Description
    IK-862 is a selective inhibitor of TACE.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    MMP
  • Recptor
    MMP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    478911-60-3
  • Formula Weight
    433.5
  • Molecular Formula
    C25H27N3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C[C@@]1(C(=O)N([C@@H](C(NO)=O)C)CC1)C2=CC=C(OCC=3C4=C(N=C(C)C3)C=CC=C4)C=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Georgiadis D, et al. Specific targeting of metzincin family members with small-molecule inhibitors: progress toward a multifarious challenge. Bioorg Med Chem. 2008;16(19):8781-8794. doi:10.1016/j.bmc.2008.08.058?
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