Methyltetrazine-Amine

CAS No. 1345955-28-3

Methyltetrazine-Amine( —— )

Catalog No. M33701 CAS No. 1345955-28-3

Methyltetrazine-Amine is a methyl-substituted tetrazine amine used in the synthesis of PROTAC molecules.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 40 In Stock
25MG 77 In Stock
50MG 120 In Stock
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Biological Information

  • Product Name
    Methyltetrazine-Amine
  • Note
    Research use only, not for human use.
  • Brief Description
    Methyltetrazine-Amine is a methyl-substituted tetrazine amine used in the synthesis of PROTAC molecules.
  • Description
    Methyltetrazine-Amine, a tetrazine compound, is used for the site-specific dual functionalization of the resulting bioconjugates.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    PROTACs
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1345955-28-3
  • Formula Weight
    201.23
  • Molecular Formula
    C10H11N5
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 20.83 mg/mL (103.51 mM; ultrasonic and warming and adjust pH to 2 with HCl and heat to 60°C; )
  • SMILES
    N=1N=C(N=NC1C=2C=CC(=CC2)CN)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Antoine Maruani, et al. A Plug-and-Play Approach for the De Novo Generation of Dually Functionalized Bispecifics. Bioconjug Chem. 2020 Mar 18;31(3):520-529.?
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