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CHR-6494
CAS No. 1333377-65-3
CHR-6494( —— )
Catalog No. M33318 CAS No. 1333377-65-3
CHR-6494 is a haspin inhibitor that inhibits histone H3T3 phosphorylation (IC50: 2 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 55 | In Stock |
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| 5MG | 49 | In Stock |
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| 10MG | 75 | In Stock |
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| 25MG | 148 | In Stock |
|
| 50MG | 268 | In Stock |
|
| 100MG | 456 | In Stock |
|
| 200MG | 665 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCHR-6494
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NoteResearch use only, not for human use.
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Brief DescriptionCHR-6494 is a haspin inhibitor that inhibits histone H3T3 phosphorylation (IC50: 2 nM).
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DescriptionCHR-6494 is a potent inhibitor of haspin, with an IC50 of 2 nM. CHR-6494 inhibits histone H3T3 phosphorylation. CHR-6494 can be used in the research of cancer.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number1333377-65-3
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Formula Weight292.34
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Molecular FormulaC16H16N6
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (171.03 mM; Ultrasonic )
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SMILESOC(=O)C(F)(F)F.CCCNc1ccc2ncc(-c3ccc4[nH]ncc4c3)n2n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Huertas D, et al. Antitumor activity of a small-molecule inhibitor of the histone kinase Haspin. Oncogene. 2012 Mar 15;31(11):1408-18.?
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