YAP/TAZ inhibitor-1

CAS No. 2093565-23-0

YAP/TAZ inhibitor-1( —— )

Catalog No. M33175 CAS No. 2093565-23-0

YAP/TAZ inhibitor-1 is a YAP/TAZ inhibitor (IC50 <0.100 μΜ) for the study of abnormal immune function and cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 1093 In Stock
2MG 463 In Stock
5MG 785 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    YAP/TAZ inhibitor-1
  • Note
    Research use only, not for human use.
  • Brief Description
    YAP/TAZ inhibitor-1 is a YAP/TAZ inhibitor (IC50 <0.100 μΜ) for the study of abnormal immune function and cancer.
  • Description
    YAP/TAZ inhibitor-1 is a YAP/TAZ inhibitor extracted from patent WO2017058716A1, Compound 1, has an IC50 of <0.100 μΜ in firefly luciferase assay.
  • In Vitro
    YAP and TAZ are transcriptional co-activators of the Hippo pathway network and regulate cell proliferation, migration, and apoptosis. YAP/TAZ inhibitor-1 is an inhibitor of transcriptional coactivator with PDZ binding motif/Yes- associated protein transcriptional coactivator (TAZ/YAP).
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    YAP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2093565-23-0
  • Formula Weight
    621.81
  • Molecular Formula
    C33H39N3O5S2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 62.5 mg/mL (100.51 mM; Ultrasonic )
  • SMILES
    CC(N1CCN(CC1)S(=O)(=O)c1ccc2-c3ccc(cc3\C(=N/O)c2c1)S(=O)(=O)C1CCC(C)(C)CC1)c1ccccc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Tracy Tzu-Ling Tang Lin, et al. Tricyclic compounds. WO2017058716A1.
molnova catalog
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