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Temiverine hydrochloride
CAS No. 136529-33-4
Temiverine hydrochloride( —— )
Catalog No. M33143 CAS No. 136529-33-4
Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 686 | In Stock |
|
| 10MG | 938 | In Stock |
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| 25MG | 1444 | In Stock |
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| 50MG | 1841 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameTemiverine hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionTemiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.
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DescriptionTemiverine hydrochloride is a synthesized agent that is expected to have anticholinergic action. Temiverine hydrochloride is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
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In VitroAtropine (1 nM to 1 μM), Oxybutynin (10 nM to 10 μM), Temiverine (10 nM to 10 μM), and RCC-36 (10 nM to 1 μM) cause a parallel shift to the right of the concentration-response curves to acetylcholine stimulation.
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorCalcium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number136529-33-4
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Formula Weight422
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Molecular FormulaC24H36ClNO3
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.O=C(OC(C#CCN(CC)CC)(C)C)C(O)(C=1C=CC=CC1)C2CCCCC2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kikukawa H, et al.Pharmacologic actions of temiverine (p-INN) and its active metabolite, RCC-36, on isolated human urinary bladder muscle. Int J Urol. 1998 May;5(3):268-75.?
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