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(Rac)-VU 6008667
CAS No. 2092917-63-8
(Rac)-VU 6008667( —— )
Catalog No. M33096 CAS No. 2092917-63-8
(Rac)-VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 82 | Get Quote |
|
| 5MG | 141 | Get Quote |
|
| 10MG | 259 | Get Quote |
|
| 25MG | 422 | Get Quote |
|
| 50MG | 623 | Get Quote |
|
| 100MG | 867 | Get Quote |
|
| 500MG | 1737 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product Name(Rac)-VU 6008667
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NoteResearch use only, not for human use.
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Brief Description(Rac)-VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.
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Description(Rac)-VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetAChR
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RecptorAChR
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Research Area——
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Indication——
Chemical Information
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CAS Number2092917-63-8
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Formula Weight438.85
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Molecular FormulaC24H17ClF2N2O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC(=O)(N1C2(C=3C(C(=O)N2CC1)=CC=CC3)C4=CC(C)=C(Cl)C=C4)C5=CC(F)=C(F)C=C5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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