Cart
sales@molnova.com
Deriglidole
CAS No. 122830-14-2
Deriglidole( —— )
Catalog No. M32880 CAS No. 122830-14-2
Deriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 451 | In Stock |
|
| 5MG | 604 | In Stock |
|
| 10MG | 809 | In Stock |
|
| 25MG | 1197 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameDeriglidole
-
NoteResearch use only, not for human use.
-
Brief DescriptionDeriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors.
-
DescriptionDeriglidole is a peripheral adrenoceptor antagonist with a high affinity for α2-adrenoceptors.
-
In VitroDeriglidole is a selective α2-receptor inhibitor. Deriglidole inhibits [3H]Clonidine and [3H]Idazoxan but not [3H]Prazosin binding to rat cortical and human platelet α2-adrenoceptors and is more selective than Idazoxan for peripheral receptors.
-
In Vivo——
-
Synonyms——
-
PathwayGPCR/G Protein
-
TargetAdrenergic Receptor
-
RecptorAdrenergic Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number122830-14-2
-
Formula Weight255.36
-
Molecular FormulaC16H21N3
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC(CC)C1(N2C=3C(C1)=CC=CC3CC2)C=4NCCN4
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Natali A,et al. Effects of acute alpha 2-blockade on insulin action and secretion in humans. Am J Physiol. 1998 Jan;274(1 Pt 1):E57-64.?
molnova catalog
related products
-
JP1302
JP1302 is a selective α2C adrenoceptor antagonist with a Kb value of 16 nM and a Ki of 28 nM for human α2C receptors.
-
Acebutolol hydrochlo...
A cardioselective beta blocker for the treatment of hypertension and arrhythmias.
-
BODIPY FL prazosin
BODIPY FL prazosin is a fluorescent α1-adrenergic antagonist with binding affinities of Ki: 14.5 nM for α1a-AR and Ki: 43.3 nM for α1b-AR, used to study subcellular localization differences in α1-adrenoceptor subtypes.
