Epsilon-momfluorothrin (Momfluorothrin, (Z,1R,3R)-), a type I synthetic pyrethroid insecticide, exerts its insecticidal properties and triggers activation of the constitutive androstane receptor (CAR).

UV0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).

Coumaperine, a product found in white pepper, is also a 5-LOX inhibitor with potential anti-inflammatory and anti-cancer activity and can be used to study inflammatory diseases caused by bacterial infections.