Gymnemagenin is a potent and selective antagonist for the β isoform of LXR it has antihyperglycemic activity.

FM1-43 is a highly lipophilic, water-soluble styrene dye that acts as an osmotic blocker of hair cell mechanical transducer channels and can be used to study neuropeptide granule dynamics and cytotoxicity.

XY101 is a selective, metabolically stable and orally available agonist of RORγ inverse(IC50 of 30 nM and a Kd of 380 nM).