Elevenostat
CAS No. 1454902-97-6
Elevenostat( JB3-22 )
Catalog No. M28876 CAS No. 1454902-97-6
Elevenostat is an HDAC11-selective inhibitor with an IC50 value of 0.235 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 35 | In Stock |
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| 10MG | 58 | In Stock |
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| 25MG | 110 | In Stock |
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| 50MG | 177 | In Stock |
|
| 100MG | 330 | In Stock |
|
| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameElevenostat
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NoteResearch use only, not for human use.
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Brief DescriptionElevenostat is an HDAC11-selective inhibitor with an IC50 value of 0.235 μM.
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DescriptionElevenostat is an HDAC11-selective inhibitor with an IC50 value of 0.235 μM.(In Vitro):Elevenostat induced cell death in MM cell lines.(In Vivo):Elevenostat produced similar anti-MM activity in vivo, improving survival among mice inoculated with 5TGM1 MM cells.
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In Vitro——
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In Vivo——
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SynonymsJB3-22
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorTelomerase
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Research Area——
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Indication——
Chemical Information
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CAS Number1454902-97-6
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Formula Weight315.32
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Molecular FormulaC16H17N3O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (792.85 mM)
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SMILESCOc(cccc1)c1NC(NCc(cc1)ccc1C(NO)=O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Fleming AM, et al. Human DNA Repair Genes Possess Potential G-Quadruplex Sequences in Their Promoters and 5'-Untranslated Regions. Biochemistry. 2018 Feb 13;57(6):991-1002.
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