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Stafia-1
CAS No. 2582757-90-0
Stafia-1( —— )
Catalog No. M28612 CAS No. 2582757-90-0
Stafia-1 is a potent STAT5a inhibitor ( IC50=22.2 μM). Stafia-1 displays high selectivity over STAT5b and other STAT family members.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 218 | In Stock |
|
| 5MG | 187 | In Stock |
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| 10MG | 310 | In Stock |
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| 25MG | 525 | In Stock |
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| 50MG | 740 | In Stock |
|
| 100MG | 1014 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 2065 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameStafia-1
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NoteResearch use only, not for human use.
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Brief DescriptionStafia-1 is a potent STAT5a inhibitor ( IC50=22.2 μM). Stafia-1 displays high selectivity over STAT5b and other STAT family members.
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DescriptionStafia-1 is a potent STAT5a inhibitor ( IC50=22.2 μM). Stafia-1 displays high selectivity over STAT5b and other STAT family members.
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In VitroStafia-1 shows at least 9-fold selectivity over STAT5b and higher selectivity against other STAT family members.
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In Vivo——
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Synonyms——
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PathwayJAK/STAT Signaling
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TargetSTAT
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RecptorNOP receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2582757-90-0
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Formula Weight506.44
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Molecular FormulaC24H27O10P
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (493.64 mM)
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SMILESCOC1=CC(C2=CC(OP(O)(O)=O)=CC(C3=CC(OC)=C(OC)C(OC)=C3)=C2)=CC(OC)=C1OC
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Thomsen C, Hohlweg R. (8-Naphthalen-1-ylmethyl-4-oxo-1-phenyl-1,3,8-triaza-spiro[4. 5]dec-3-yl)-acetic acid methyl ester (NNC 63-0532) is a novel potent nociceptin receptor agonist. Br J Pharmacol. 2000 Nov;131(5):903-8.
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