A2B receptor antagonist 2

CAS No. 784-90-7

A2B receptor antagonist 2( —— )

Catalog No. M28147 CAS No. 784-90-7

A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
25MG 57 Get Quote
50MG 83 Get Quote
100MG Get Quote Get Quote
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Biological Information

  • Product Name
    A2B receptor antagonist 2
  • Note
    Research use only, not for human use.
  • Brief Description
    A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
  • Description
    A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Apoptosis
  • Target
    Adenosine Receptor
  • Recptor
    CD11b
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    784-90-7
  • Formula Weight
    229.287
  • Molecular Formula
    C12H15N5
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 2 mg/mL (8.72 mM)
  • SMILES
    Cc1cc2nc(NC(N)=N)nc(C)c2cc1C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Panni RZ, et al. Agonism of CD11b reprograms innate immunity to sensitize pancreatic cancer to immunotherapies. Sci Transl Med. 2019 Jul 3;11(499).
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