TPX-0046

CAS No. 2359650-19-2

TPX-0046( —— )

Catalog No. M28037 CAS No. 2359650-19-2

TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 220 In Stock
5MG 353 In Stock
10MG 549 In Stock
25MG 1036 In Stock
50MG 1376 In Stock
100MG 1841 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    TPX-0046
  • Note
    Research use only, not for human use.
  • Brief Description
    TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.
  • Description
    TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    p97
  • Recptor
    BCRP|ABCG2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2359650-19-2
  • Formula Weight
    424.43
  • Molecular Formula
    C21H21FN6O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C1NC[C@@H](C)OC2=NC=C(F)C=C2CN3C4=NC5=C1C=NN5C=C4O[C@@]6([H])[C@]3([H])CCC6
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Milligan SR, et al. The endocrine activities of 8-prenylnaringenin and related hop (Humulus lupulus L.) flavonoids. J Clin Endocrinol Metab. 2000 Dec;85(12):4912-5.
molnova catalog
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