Suprafenacine

CAS No. 1477482-50-0

Suprafenacine( N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide )

Catalog No. M27928 CAS No. 1477482-50-0

Suprafenacine is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 199 Get Quote
10MG 282 Get Quote
25MG 507 Get Quote
50MG 712 Get Quote
100MG 1008 Get Quote
500MG 2025 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Suprafenacine
  • Note
    Research use only, not for human use.
  • Brief Description
    Suprafenacine is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase.
  • Description
    Suprafenacine is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase. Suprafenacine binds to microtubules and inhibits aggregation at the colchicine junction. Suprafenacine is selective for cancer cells, including drug-resistant cancer cells.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    Microtubule/Tubulin
  • Recptor
    β2-adrenergic receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1477482-50-0
  • Formula Weight
    282.347
  • Molecular Formula
    C16H18N4O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cc1ccc(\C=N\NC(=O)c2n[nH]c3CCCCc23)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Shuyun Bi, et al. Study on the interactions of mapenterol with serum albumins using multi-spectroscopy and molecular docking. Luminescence. 2016 Mar;31(2):372-379.
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