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DDD85646

CAS No. 1215010-55-1

DDD85646( DDD-85646 | DDD 85646 )

Catalog No. M27869 CAS No. 1215010-55-1

DDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 284 Get Quote
10MG 442 Get Quote
25MG 645 Get Quote
50MG 896 Get Quote
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Biological Information

  • Product Name
    DDD85646
  • Note
    Research use only, not for human use.
  • Brief Description
    DDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.
  • Description
    DDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    DDD-85646 | DDD 85646
  • Pathway
    Microbiology/Virology
  • Target
    Parasite
  • Recptor
    GABAA
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1215010-55-1
  • Formula Weight
    495.42
  • Molecular Formula
    C21H24Cl2N6O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (201.84 mM)
  • SMILES
    Cc1nn(C)c(C)c1NS(=O)(=O)c1c(Cl)cc(cc1Cl)-c1ccnc(c1)N1CCNCC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Quan Z, et al. Reactive oxygen species-mediated endoplasmic reticulum stress and mitochondrial dysfunction contribute to cirsimaritin-induced apoptosis in human gallbladder carcinoma GBC-SD cells. Cancer Lett. 2010 Sep 28;295(2):252-9.
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