CAY10526( CAY-10526 | CAY 10526 | BTH )

Catalog No. M27762 CAS No. 938069-71-7

CAY10526 is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

CAY10526
Note

Research use only, not for human use.
Brief Description

CAY10526 is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.
Description

CAY10526 is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.(In Vitro):CAY10526 dose-dependently inhibits PGE2 production in lipopolysaccharide-stimulated RAW 264.7 cells with an IC50 value of 1.8 μM without any effect on COX-2 expression.
In Vitro

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In Vivo

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Synonyms

CAY-10526 | CAY 10526 | BTH
Pathway

GPCR/G Protein
Target

Prostaglandin Receptor
Recptor

CDK
Research Area

——
Indication

——

Chemical Information

CAS Number

938069-71-7
Formula Weight

311.15
Molecular Formula

C12H7BrO3S
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 66.67 mg/mL (214.27 mM)
SMILES

OC1OC(=O)C(Br)=C1c1cc2ccccc2s1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Tadesse S, Zhu G, Mekonnen LB, Lenjisa JL, Yu M, Brown MP, Wang S. A novel series of N-(pyridin-2-yl)-4-(thiazol-5-yl)pyrimidin-2-amines as highly potent CDK4/6 inhibitors. Future Med Chem. 2017 Sep;9(13):1495-1506.

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