Remoxipride hydrochloride

CAS No. 73220-03-8

Remoxipride hydrochloride( Roxiam | (S)-Remoxipride Hydrochloride | Remoxipride Hydrochloride Anhydrous )

Catalog No. M27695 CAS No. 73220-03-8

Dopamine D2 receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 85 In Stock
10MG 132 In Stock
25MG 264 In Stock
50MG 390 In Stock
100MG 576 In Stock
200MG Get Quote In Stock
500MG 1190 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Remoxipride hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Dopamine D2 receptor antagonist.
  • Description
    Dopamine D2 receptor antagonist.(In Vivo):In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting.
  • In Vitro
    (S)-Remoxipride hydrochloride (1-100 μM; 20 min) shows binding efficiency with IC50s of >100, 1.57 and 42 μM for dopamine D1, dopamine D2 and α1-Adrenoccptor, respectively.
  • In Vivo
    (S)-Remoxipride hydrochloride (0.1-100 μM/kg; i.p. 60 min prior to apomorphine) blockades apomorphine-induced behaviors s in rats and vomiting in dogs.(S)-Remoxipride hydrochloride (0.1-10 mg/kg; i.p. 30 min prior to apomorphine) displaces [3H]spiperone from both striatal and extra-striatal areas.
  • Synonyms
    Roxiam | (S)-Remoxipride Hydrochloride | Remoxipride Hydrochloride Anhydrous
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    73220-03-8
  • Formula Weight
    407.73
  • Molecular Formula
    C16H24BrClN2O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.CCN1CCC[C@H]1CNC(=O)c1c(OC)ccc(Br)c1OC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Richard W. Watkins, et al. Evaluation of cinnamamide as an avian repellent: Determination of a dose—response curve.
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