PNU-177864

CAS No. 250266-51-4

PNU-177864( —— )

Catalog No. M27686 CAS No. 250266-51-4

dopamine D3 receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 72 In Stock
10MG 89 In Stock
25MG 202 In Stock
50MG 277 In Stock
100MG 383 In Stock
200MG 533 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PNU-177864
  • Note
    Research use only, not for human use.
  • Brief Description
    dopamine D3 receptor antagonist.
  • Description
    dopamine D3 receptor antagonist.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Male and female Sprague-Dawley rats (8-9-week-old)Dosage:12.5 mg/kg, 50 mg/kg (for 2 weeks), or 200 mg/kg; 8 mg/kg, 25 mg/kg, or 80 mg/kg (for 4 weeks)Administration:Oral gavage; daily; for 2-4 weeksResult:Induced phospholipidosis in unusual target organs in dogs or rats including epididymis, pituitary, and hair follicles.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    PI3K|Caspase|Bcl-2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    250266-51-4
  • Formula Weight
    438.89
  • Molecular Formula
    C18H21F3N2O3S·HCl
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCCNCCC1=CC=C(NS(C2=CC=C(OC(F)(F)F)C=C2)(=O)=O)C=C1.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Tomonaga T, et al. Isoflavonoids, genistein, psi-tectorigenin, and orobol, increase cytoplasmic free calcium in isolated rat hepatocytes. Biochem Biophys Res Commun. 1992 Jan 31;182(2):894-9.
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