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Ocinaplon
CAS No. 96604-21-6
Ocinaplon( DOV 273547 )
Catalog No. M27674 CAS No. 96604-21-6
Ocinaplon is a GABAA receptors modulator.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 80 | Get Quote |
|
| 10MG | 140 | Get Quote |
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| 25MG | 282 | Get Quote |
|
| 50MG | 421 | Get Quote |
|
| 100MG | 606 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameOcinaplon
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NoteResearch use only, not for human use.
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Brief DescriptionOcinaplon is a GABAA receptors modulator.
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DescriptionOcinaplon is a GABAA receptors modulator.(In Vivo):In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test.
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In Vitro——
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In Vivo——
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SynonymsDOV 273547
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PathwayOthers
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TargetOther Targets
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RecptorP2X7
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Research Area——
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Indication——
Chemical Information
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CAS Number96604-21-6
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Formula Weight301.309
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Molecular FormulaC17H11N5O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 2 mg/mL (6.64 mM)
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SMILESO=C(c1cnn2c(ccnc12)-c1ccncc1)c1ccccn1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Hopper AT, et al. Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139. J Med Chem. 2021;64(8):4891-4902.
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