L-838417 D9

CAS No. 1213669-91-0

L-838417 D9( CTP354 | C-21191 )

Catalog No. M27542 CAS No. 1213669-91-0

L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 53 In Stock
2MG 29 In Stock
5MG 44 In Stock
10MG 65 In Stock
25MG 130 In Stock
50MG 207 In Stock
100MG 333 In Stock
200MG 462 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    L-838417 D9
  • Note
    Research use only, not for human use.
  • Brief Description
    L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes.
  • Description
    L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CTP354 | C-21191
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    TFIIH
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1213669-91-0
  • Formula Weight
    408.45
  • Molecular Formula
    C19H19F2N7O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 12.5 mg/mL (30.60 mM)
  • SMILES
    CN1N=CN=C1COC2=NN3C(C=C2C(C([2H])([2H])[2H])(C([2H])([2H])[2H])C([2H])([2H])[2H])=NN=C3C4=CC(F)=CC=C4F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Pinho-Ribeiro FA, et al. Protective effects of the flavonoid hesperidin methyl chalcone in inflammation and pain in mice: role of TRPV1, oxidative stress, cytokines and NF-κB. Chem Biol Interact. 2015 Feb 25;228:88-99.
molnova catalog
related products
  • 4-Methylkaempferol

    4'-Methylkaempferol

  • Flavanone

    Used as organic synthesis and medicine intermediate.

  • 5-HT2B antagonist-1

    5-HT2B antagonist-1 is an orally active 5-HT2B receptor antagonist with an IC50 of 33.4 nM, suitable for studies of diseases characterized by 5-HT2B receptor signaling, such as hepatocellular carcinoma, cardiovascular disease, or gastrointestinal disease .