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AZ 11645373
CAS No. 227088-94-0
AZ 11645373( 3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE )
Catalog No. M27445 CAS No. 227088-94-0
AZ 11645373 is a highly selective and potent human P2X7 receptor antagonist that has no effect on mouse/rat P2X7 receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 107 | In Stock |
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| 5MG | 103 | In Stock |
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| 10MG | 148 | In Stock |
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| 25MG | 250 | In Stock |
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| 50MG | 346 | In Stock |
|
| 100MG | 483 | In Stock |
|
| 200MG | 643 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAZ 11645373
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NoteResearch use only, not for human use.
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Brief DescriptionAZ 11645373 is a highly selective and potent human P2X7 receptor antagonist that has no effect on mouse/rat P2X7 receptor.
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DescriptionAZ 11645373 is a highly selective and potent human P2X7 receptor antagonist that has no effect on mouse/rat P2X7 receptor.
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In Vitro——
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In Vivo——
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Synonyms3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE
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PathwayMembrane Transporter/Ion Channel
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TargetP2X Receptor
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number227088-94-0
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Formula Weight463.51
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Molecular FormulaC24H21N3O5S
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Purity>98% (HPLC)
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Solubility——
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SMILES[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccncc2)N2C(=O)CSC2=O)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Qiao-yu Yuan,et al. Chemical Constituents from Cremastra appendiculata. Zhong Yao Cai. 2015 Feb;38(2):298-301.
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