Varespladib methyl

CAS No. 172733-08-3

Varespladib methyl( A-002 | LY333013 )

Catalog No. M26858 CAS No. 172733-08-3

Varespladib methyl, a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 233 In Stock
2MG 125 In Stock
5MG 211 In Stock
10MG 337 In Stock
25MG 558 In Stock
50MG 754 In Stock
100MG 1032 In Stock
200MG 1376 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Varespladib methyl
  • Note
    Research use only, not for human use.
  • Brief Description
    Varespladib methyl, a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.
  • Description
    Varespladib methyl, a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor. (In Vitro):Varespladib methyl display high-level secretory PLA2 inhibition at nanomolar and picomolar concentrations against 28 medically important snake venoms from six continents .
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    A-002 | LY333013
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Endogenous Metabolite
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    172733-08-3
  • Formula Weight
    394.427
  • Molecular Formula
    C22H22N2O5
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (253.54 mM)
  • SMILES
    CCc1c(C(=O)C(N)=O)c2c(OCC(=O)OC)cccc2n1Cc1ccccc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Morley SR, Forrest AR, Galloway JH. Validation of meconin as a marker for illicit opiate use. J Anal Toxicol. 2007 Mar;31(2):105-8.
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