DGAT1-IN-1( —— )

Catalog No. M26665 CAS No. 1449779-49-0

DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

DGAT1-IN-1
Note

Research use only, not for human use.
Brief Description

DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).
Description

DGAT1-IN-1 is a potent inhibitor of diacylglycerol O- acyltransferase type 1(DGAT1, IC50 of < 10 nM).(In Vitro):Various concentrations (0.0008 μΜ, 0.004 μΜ, 0.02 μΜ, 0.1 μΜ, 0.5 μΜ, 2.5 μΜ and 10.0 μΜ) of the compounds of Examples were added to individual wells prior to the addition of the cell lysates, or human or mouse liver microsomes.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Metabolic Enzyme/Protease
Target

Transferase
Recptor

Centromere-Associated Protein E
Research Area

——
Indication

——

Chemical Information

CAS Number

1449779-49-0
Formula Weight

551.566
Molecular Formula

C30H28F3N3O4
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 20 mg/mL (36.26 mM)
SMILES

OC(=O)C[C@H]1CC[C@@H](CC1)c1ccc(cc1)-c1ccc2nc(cn2c1)C(=O)NCc1ccc(OC(F)(F)F)cc1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Qian X, et al. Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295. ACS Med Chem Lett. 2010 Jan 19;1(1):30-4.

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