CCG-63808( —— )

Catalog No. M26641 CAS No. 620113-73-7

CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

CCG-63808
Note

Research use only, not for human use.
Brief Description

CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.
Description

CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. CCG-63808 dose-dependently inhibits the TR-FRET signal between RGS4-AF488 and Tb-Gαo with IC50 values of 1.9 μM.(In Vitro):CCG-63808 showed selectivity among RGS proteins with a potency order of RGS 4 > 19 = 16 > 8 7. CCG-63808 inhibited the GTPase accelerating protein activity of RGS4.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

melanocortin 3 (MC3)| melanocortin-1 receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

620113-73-7
Formula Weight

454.48
Molecular Formula

C25H15FN4O2S
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 1 mg/mL (2.20 mM)
SMILES

Cc1cccn2c1nc(Oc1ccc(F)cc1)c(\C=C(/C#N)c1nc3ccccc3s1)c2=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Montero-Melendez T, et al. Biased agonism as a novel strategy to harness the proresolving properties of melanocortin receptors without eliciting melanogenic effects. J Immunol. 2015 Apr 1;194(7):3381-8.

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