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Rho-Kinase-IN-1
CAS No. 1035094-83-7
Rho-Kinase-IN-1( —— )
Catalog No. M26415 CAS No. 1035094-83-7
Rho-Kinase-IN-1 is a inhibitor of Rho kinase (ROCK) with Ki values of 30.5 and 3.9 nM for ROCK1 and ROCK2, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 107 | In Stock |
|
| 5MG | 141 | In Stock |
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| 10MG | 216 | In Stock |
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| 25MG | 377 | In Stock |
|
| 50MG | 518 | In Stock |
|
| 100MG | 686 | In Stock |
|
| 200MG | 923 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRho-Kinase-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionRho-Kinase-IN-1 is a inhibitor of Rho kinase (ROCK) with Ki values of 30.5 and 3.9 nM for ROCK1 and ROCK2, respectively.
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DescriptionRho-Kinase-IN-1 is a inhibitor of Rho kinase (ROCK) with Ki values of 30.5 and 3.9 nM for ROCK1 and ROCK2, respectively.
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In VitroRho-Kinase-IN-1 is a ROCK inhibitor which can be useful for treating diseases or conditions associated with excessive cell proliferation, remodeling, edema and inflammation.
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetROCK
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RecptorCaspase| PAFR| PARP
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Research Area——
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Indication——
Chemical Information
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CAS Number1035094-83-7
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Formula Weight352.5
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Molecular FormulaC20H24N4S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (141.84 mM)
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SMILESCSc1ccc(CN2CCCC(C2)Nc2ccc3[nH]ncc3c2)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Wang JJ, Liu YX, et al. [Study on steroidal saponins from Dioscorea zingiberensis and their platelet aggregation activities]. Zhongguo Zhong Yao Za Zhi. 2014 Oct;39(19):3782-7. Chinese.
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