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Pinacidil
CAS No. 60560-33-0
Pinacidil( P-1134 | P 1134 | P1134 | S-1230 | S 1230 )
Catalog No. M26377 CAS No. 60560-33-0
Pinardil (P-1134, S-1230) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and peripheral resistance and producing fluid retention.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 44 | In Stock |
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| 5MG | 40 | In Stock |
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| 10MG | 55 | In Stock |
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| 25MG | 92 | In Stock |
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| 50MG | 153 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePinacidil
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NoteResearch use only, not for human use.
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Brief DescriptionPinardil (P-1134, S-1230) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and peripheral resistance and producing fluid retention.
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DescriptionPinardil (P-1134, S-1230) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and peripheral resistance and producing fluid retention.
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In Vitro——
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In Vivo——
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SynonymsP-1134 | P 1134 | P1134 | S-1230 | S 1230
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PathwayCell Cycle/DNA Damage
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TargetPotassium Channel
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RecptorFatty Acid Synthase (FASN)
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Research Area——
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Indication——
Chemical Information
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CAS Number60560-33-0
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Formula Weight245.33
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Molecular FormulaC13H19N5
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (407.63 mM)
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SMILESCC(C)(C)C(N/C(NC1=CC=NC=C1)=N/C#N)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Alwarawrah Y, Hughes P, Loiselle D, Carlson DA, Darr DB, Jordan JL, Xiong J, Hunter LM, Dubois LG, Thompson JW, Kulkarni MM, Ratcliff AN, Kwiek JJ, Haystead TA. Fasnall, a Selective FASN Inhibitor, Shows Potent Anti-tumor Activity in the MMTV-Neu Model of HER2(+) Breast Cancer. Cell Chem Biol. 2016 Jun 23;23(6):678-88.
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