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PD 168568 dihydrochloride

CAS No. 1782532-06-2

PD 168568 dihydrochloride( PD 168568 (dihydrochloride) )

Catalog No. M26360 CAS No. 1782532-06-2

PD 168568 dihydrochloride is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PD 168568 dihydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    PD 168568 dihydrochloride is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
  • Description
    PD 168568 dihydrochloride is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).(In Vitro):PD 168568 dihydrochloride has good selective for D4 receptor(Ki of 1842 nM for D2 receptor).(In Vivo):PD 168568 dihydrochloride inhibit amphetamine stimulated locomotor activity in the rat.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Rat Dosage:3 mg/kg Administration:Oral administration Result:Inhibit amphetamine (0.5 mg/kg, i.p.) stimulated locomotor activity.
  • Synonyms
    PD 168568 (dihydrochloride)
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    α4β2 nAChR| α7 nAChR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1782532-06-2
  • Formula Weight
    422.39
  • Molecular Formula
    C22H29Cl2N3O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.Cl.Cc1ccc(cc1C)N1CCN(CCC2NC(=O)c3ccccc23)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Stevens KE, Kem WR, Mahnir VM, Freedman R. Selective alpha7-nicotinic agonists normalize inhibition of auditory response in DBA mice. Psychopharmacology (Berl). 1998 Apr;136(4):320-7.
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