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Home - Products - Metabolic Enzyme/Protease - P450 - N-Desmethyl-Apalutamide

N-Desmethyl-Apalutamide

CAS No. 1332391-11-3

N-Desmethyl-Apalutamide( N-Desmethyl Apalutamide )

Catalog No. M26314 CAS No. 1332391-11-3

N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 278 In Stock
5MG 259 In Stock
10MG 373 In Stock
25MG 562 In Stock
50MG 759 In Stock
100MG 1014 In Stock
200MG 1376 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    N-Desmethyl-Apalutamide
  • Note
    Research use only, not for human use.
  • Brief Description
    N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
  • Description
    N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    N-Desmethyl Apalutamide
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    P450
  • Recptor
    CYP2C9| HIV
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1332391-11-3
  • Formula Weight
    463.41
  • Molecular Formula
    C20H13F4N5O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (215.79 mM)
  • SMILES
    NC(=O)c1ccc(cc1F)N1C(=S)N(C(=O)C11CCC1)c1cnc(C#N)c(c1)C(F)(F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Chen DF, et al. Anti-AIDS agents--XXVI. Structure-activity correlations of gomisin-G-related anti-HIV lignans from Kadsura interior and of related synthetic analogues. Bioorg Med Chem. 1997 Aug;5(8):1715-23.
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