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HA155
CAS No. 1312201-00-5
HA155( CS-963 )
Catalog No. M26244 CAS No. 1312201-00-5
HA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 67 | In Stock |
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| 5MG | 65 | In Stock |
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| 10MG | 103 | In Stock |
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| 25MG | 211 | In Stock |
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| 50MG | 332 | In Stock |
|
| 100MG | 491 | In Stock |
|
| 200MG | 702 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameHA155
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NoteResearch use only, not for human use.
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Brief DescriptionHA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.
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DescriptionHA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.(In Vitro):HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA dose-dependently .HA155 is an ATX inhibitor by binding to the ATX active site .
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In VitroHA-155 inhibits ATX by binding to the ATX active site.HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA in a dose-dependent manner.
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In Vivo——
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SynonymsCS-963
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PathwayAngiogenesis
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TargetPDE
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RecptorAntibacterial
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Research Area——
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Indication——
Chemical Information
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CAS Number1312201-00-5
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Formula Weight463.29
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Molecular FormulaC24H19BFNO5S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 10 mg/mL (21.58 mM)
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SMILESO=C1N(CC2=CC=C(F)C=C2)C(S/C1=C\C3=CC=C(OCC4=CC=C(B(O)O)C=C4)C=C3)=O.[(Z)]
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Guo B, et al. Clinical Pharmacokinetics of Levornidazole in Elderly Subjects and Dosing Regimen Evaluation Using Pharmacokinetic/Pharmacodynamic Analysis. Clin Ther. 2017 Jul;39(7):1336-1346.
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