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Lenacapavir
CAS No. 2189684-44-2
Lenacapavir( GS-6207 )
Catalog No. M26233 CAS No. 2189684-44-2
Lenacapavir is a potent capsid-targeting inhibitor of HIV replication. Lenacapavir shows anti-HIV activity with an EC50 of 100 pM in MT-4 cells.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 616 | In Stock |
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| 5MG | 376 | In Stock |
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| 10MG | 565 | In Stock |
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| 25MG | 998 | In Stock |
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| 50MG | 1358 | In Stock |
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| 100MG | 1841 | In Stock |
|
| 200MG | 2567 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLenacapavir
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NoteResearch use only, not for human use.
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Brief DescriptionLenacapavir is a potent capsid-targeting inhibitor of HIV replication. Lenacapavir shows anti-HIV activity with an EC50 of 100 pM in MT-4 cells.
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DescriptionLenacapavir is a potent capsid-targeting inhibitor of HIV replication. Lenacapavir shows anti-HIV activity with an EC50 of 100 pM in MT-4 cells.(In Vitro):Lenacapavir displays a mean EC50 of 50 pM (20-160 pM) against 23 HIV-1 clinical isolates from different subtypes in peripheral blood mononuclear cells. Lenacapavir shows sub-nanomolar potency in target cells with EC50 of 23 pM, in a full-cycle assay with EC50 of 25 pM and in producer cells with EC50 of 439 pM.
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In Vitro——
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In Vivo——
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SynonymsGS-6207
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PathwayOthers
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TargetOther Targets
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number2189684-44-2
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Formula Weight968.28
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Molecular FormulaC39H32ClF10N7O5S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 200 mg/mL (206.55 mM)
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SMILES[H][C@]12C[C@@]1([H])C(F)(F)c1c2c(nn1CC(=O)N[C@@H](Cc1cc(F)cc(F)c1)c1nc(ccc1-c1ccc(Cl)c2c(NS(C)(=O)=O)nn(CC(F)(F)F)c12)C#CC(C)(C)S(C)(=O)=O)C(F)(F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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