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3-Bromocytisine

CAS No. 207390-14-5

3-Bromocytisine( 3-Br-cytisine | (-)-3-Bromocytisine | (-)-9-Bromocytisine )

Catalog No. M26025 CAS No. 207390-14-5

3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 188 In Stock
5MG 214 In Stock
10MG 309 In Stock
25MG 521 In Stock
50MG 733 In Stock
100MG 1004 In Stock
200MG 1349 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    3-Bromocytisine
  • Note
    Research use only, not for human use.
  • Brief Description
    3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).
  • Description
    3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).(In Vitro):3-Bromocytisine shows different effects on high and low ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively .
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    3-Br-cytisine | (-)-3-Bromocytisine | (-)-9-Bromocytisine
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    D4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    207390-14-5
  • Formula Weight
    269.142
  • Molecular Formula
    C11H13BrN2O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (371.55 mM)
  • SMILES
    Brc1ccc2[C@H]3CNC[C@H](C3)Cn2c1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Nakazawa S, et al. Behavioral and neurophysiological effects of Ro 10-5824, a dopamine D4 receptor partial agonist, in common marmosets. Psychopharmacology (Berl). 2015 Sep;232(17):3287-95.
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