EP1-antagonist-1

CAS No. 851204-35-8

EP1-antagonist-1( EP1 antagonist 1 )

Catalog No. M26017 CAS No. 851204-35-8

EP1-antagonist-1 is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 256 In Stock
5MG 226 In Stock
10MG 330 In Stock
25MG 520 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    EP1-antagonist-1
  • Note
    Research use only, not for human use.
  • Brief Description
    EP1-antagonist-1 is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
  • Description
    EP1-antagonist-1 is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    EP1 antagonist 1
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Cleavable
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    851204-35-8
  • Formula Weight
    470.14
  • Molecular Formula
    C19H15BrCl2N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cc1cc(nn1Cc1cc(Br)ccc1OCc1ccc(Cl)cc1Cl)C(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Staben LR, et al. Stabilizing a Tubulysin Antibody-Drug Conjugate To Enable Activity Against Multidrug-Resistant Tumors. ACS Med Chem Lett. 2017 Sep 5;8(10):1037-1041.
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