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Vanilloid receptor antagonist 1

CAS No. 871814-52-7

Vanilloid receptor antagonist 1( 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile )

Catalog No. M24886 CAS No. 871814-52-7

Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 37 In Stock
5MG 235 In Stock
10MG 353 In Stock
25MG 601 In Stock
50MG 830 In Stock
100MG 1181 In Stock
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Biological Information

  • Product Name
    Vanilloid receptor antagonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
  • Description
    Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPV1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    871814-52-7
  • Formula Weight
    305.33
  • Molecular Formula
    C18H15N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (327.51 mM)
  • SMILES
    CC(C)C(N1c(cc2)ccc2C#N)=Nc(cc(cc2)O)c2C1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ritchie T J , Culshaw A J , Brain C T , et al. Quinazolinone derivatives useful as vanilloid antagonists: US, US8349852 B2[P]. 2012.
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