Vanilloid receptor antagonist 1

CAS No. 871814-52-7

Vanilloid receptor antagonist 1( 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile )

Catalog No. M24886 CAS No. 871814-52-7

Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 37 In Stock
5MG 235 In Stock
10MG 353 In Stock
25MG 601 In Stock
50MG 830 In Stock
100MG 1181 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Vanilloid receptor antagonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
  • Description
    Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPV1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    871814-52-7
  • Formula Weight
    305.33
  • Molecular Formula
    C18H15N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (327.51 mM)
  • SMILES
    CC(C)C(N1c(cc2)ccc2C#N)=Nc(cc(cc2)O)c2C1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ritchie T J , Culshaw A J , Brain C T , et al. Quinazolinone derivatives useful as vanilloid antagonists: US, US8349852 B2[P]. 2012.
molnova catalog
related products
  • N-Oleoyl Glutamine

    N-Oleoyl Glutamine (Oleoyl-L-glutamine) is an N-acyl amino acid involved in the regulation of PM20D1 and antagonizes TRPV1 of the transient receptor potential (TRP) calcium channel.

  • ASP7663

    ASP7663 is a?TRPA1 Receptor Agonist?and exhibiting an abdominal analgesic effect in vivo.?

  • AM-0902

    AM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).