Vanilloid receptor antagonist 1

CAS No. 871814-52-7

Vanilloid receptor antagonist 1( 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile )

Catalog No. M24886 CAS No. 871814-52-7

Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 37 In Stock
5MG 235 In Stock
10MG 353 In Stock
25MG 601 In Stock
50MG 830 In Stock
100MG 1181 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Vanilloid receptor antagonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
  • Description
    Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPV1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    871814-52-7
  • Formula Weight
    305.33
  • Molecular Formula
    C18H15N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (327.51 mM)
  • SMILES
    CC(C)C(N1c(cc2)ccc2C#N)=Nc(cc(cc2)O)c2C1=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ritchie T J , Culshaw A J , Brain C T , et al. Quinazolinone derivatives useful as vanilloid antagonists: US, US8349852 B2[P]. 2012.
molnova catalog
related products
  • Elismetrep

    Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.

  • Linoleoyl Ethanolami...

    Linoleoyl Ethanolamide is an endocannabinoid agent.?It acts by binding to TRPV1 increasing ERK phosphorylation and AP-1 dependent transcription in CB-receptor in an independent manner.

  • Nonivamide

    A capsaicin analog that acts as an agonist of TRPV1 channel.