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(R)-Elagolix
CAS No. 834153-87-6
(R)-Elagolix( NBI-56418 )
Catalog No. M24824 CAS No. 834153-87-6
(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 64 | In Stock |
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| 5MG | 46 | In Stock |
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| 10MG | 69 | In Stock |
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| 25MG | 140 | In Stock |
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| 50MG | 201 | In Stock |
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| 100MG | 317 | In Stock |
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| 200MG | 468 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product Name(R)-Elagolix
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NoteResearch use only, not for human use.
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Brief Description(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.
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Description(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full suppression at higher doses.
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In Vitro——
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In Vivo——
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SynonymsNBI-56418
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PathwayOthers
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TargetOther Targets
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RecptorGnRHR
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Research Area——
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Indication——
Chemical Information
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CAS Number834153-87-6
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Formula Weight631.59
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Molecular FormulaC32H30F5N3O5
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL (158.33 mM)
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SMILESCC1=C(C(=O)N(C(=O)N1CC2=C(C=CC=C2F)C(F)(F)F)C[C@@H](C3=CC=CC=C3)NCCCC(=O)O)C4=C(C(=CC=C4)OC)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Sieboldin
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Ampreloxetine hydroc...
Ampreloxetine hydrochloride (TD-9855 HCl) has anti-inflammatory activity and is a potential compound for the treatment of depression and Alzheimer's disease.
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NADH disodium salt h...
NADH is the reduced form of nicotinamide adenine dinucleotide (NAD) that can donate electrons as part of a reducing reaction. In that process NADH becomes oxidized to produce NAD+. A variety of enzymes use NADH plus H+ to reduce substrates generating NAD+ as well as the reduced product.
