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Home - Products - Endocrinology/Hormones - Opioid Receptor - [Leu5]-Enkephalin TFA(58822-25-6(free bas))

[Leu5]-Enkephalin TFA(58822-25-6(free bas))

CAS No. 73563-78-7

[Leu5]-Enkephalin TFA(58822-25-6(free bas))( Leu-enkephalin | Leucine enkephalin | Leucyl-enkephalin )

Catalog No. M24743 CAS No. 73563-78-7

[Leu5]-Enkephalin is the most potent δ-receptor ago.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 68 In Stock
10MG 45 In Stock
25MG 93 In Stock
50MG 138 In Stock
100MG 206 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    [Leu5]-Enkephalin TFA(58822-25-6(free bas))
  • Note
    Research use only, not for human use.
  • Brief Description
    [Leu5]-Enkephalin is the most potent δ-receptor ago.
  • Description
    [Leu5]-Enkephalin is the most potent δ-receptor ago.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Leu-enkephalin | Leucine enkephalin | Leucyl-enkephalin
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    δ-opioid receptor|Human Endogenous Metabolite
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    73563-78-7
  • Formula Weight
    669.64
  • Molecular Formula
    C30H38F3N5O9
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O.O=C(O)C(F)(F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Robert J Cassell , Krishna K Sharma , Hongyu Su,et al.The Meta-Position of Phe 4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors[J].Molecules, 24 (24) 2019 Dec 1
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