BMS986187( —— )

Catalog No. M24699 CAS No. 684238-37-7

BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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2MG	45	In Stock
5MG	72	In Stock
10MG	116	In Stock
25MG	227	In Stock
50MG	323	In Stock
100MG	500	In Stock
200MG	Get Quote	In Stock
500MG	1070	In Stock
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Biological Information

Product Name

BMS986187
Note

Research use only, not for human use.
Brief Description

BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
Description

BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
In Vitro

BMS-986187?(1 nM-100 uM) produces little or no activity in agonist mode, but in PAM mode (in the presence of an EC20?of leu-enkephalin (in CHO-OPRD1 cells) or endomorphin 1 (in CHO-OPRM1 cells)) produces a response with an EC50?of 48 nM in CHO-OPRD1 cells and 2?μM in CHO-OPRM1 cells.
In Vivo

——
Synonyms

——
Pathway

Endocrinology/Hormones
Target

Opioid Receptor
Recptor

δ-opioid receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

684238-37-7
Formula Weight

470.6
Molecular Formula

C31H34O4
Purity

>98% (HPLC)
Solubility

DMSO:10 mM
SMILES

CC1=CC=CC=C1COC2=CC=C(C=C2)C3C4=C(CC(CC4=O)(C)C)OC5=C3C(=O)CC(C5)(C)C
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Livingston K E , Stanczyk M A , Burford N , et al. Pharmacological Evidence for a Putative Conserved Allosteric Site on Opioid Receptors[J]. Molecular Pharmacology, 2017:mol.117.109561.

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