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AS 1269574
CAS No. 330981-72-1
AS 1269574( AS1269574 )
Catalog No. M24268 CAS No. 330981-72-1
AS 1269574 is a potent, orally available GPR119 agonist. AS1269574 has the potential for the research of type 2 diabetes.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 57 | In Stock |
|
| 2MG | 31 | In Stock |
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| 5MG | 49 | In Stock |
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| 10MG | 84 | In Stock |
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| 25MG | 168 | In Stock |
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| 50MG | 265 | In Stock |
|
| 100MG | 398 | In Stock |
|
| 200MG | 579 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAS 1269574
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NoteResearch use only, not for human use.
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Brief DescriptionAS 1269574 is a potent, orally available GPR119 agonist. AS1269574 has the potential for the research of type 2 diabetes.
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DescriptionAS 1269574 is a potent, orally available GPR119 agonist. AS1269574 has the potential for the research of type 2 diabetes.
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In Vitro——
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In VivoAS1269574 sgnificantly reduced the blood glucose AUC after 2 h (AUC0-2h) of administration. Animal Model:Eight-week-old ICR mice Dosage:100 mg/kg Administration:P.o.Result:Sgnificantly reduced the blood glucose AUC after 2 h (AUC0-2h) of administration. Similarly, plasma insulin AUC0-2h was significantly higher in the mice.
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SynonymsAS1269574
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorGPR119|TRPA1
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Research Area——
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Indication——
Chemical Information
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CAS Number330981-72-1
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Formula Weight308.18
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Molecular FormulaC13H14BrN3O
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Purity>98% (HPLC)
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SolubilityDMSO:250 mg/mL (811.24 mM; Need ultrasonic)
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SMILESCC1=CC(=NC(=N1)C2=CC=C(C=C2)Br)NCCO
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Yoshida S, et al. Identification of a novel GPR119 agonist, AS1269574, with in vitro and in vivo glucose-stimulated insulin secretion. Biochem Biophys Res Commun. 2010;400(3):437-441.
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