NVP-BHG712 isomer

CAS No. 2245892-85-5

NVP-BHG712 isomer( —— )

Catalog No. M24025 CAS No. 2245892-85-5

NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 85 In Stock
2MG 48 In Stock
5MG 76 In Stock
10MG 145 In Stock
25MG 259 In Stock
50MG 368 In Stock
100MG 548 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    NVP-BHG712 isomer
  • Note
    Research use only, not for human use.
  • Brief Description
    NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
  • Description
    NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
  • In Vitro
    NVP-BHG712 isomer exhibits IC 50 values of 163 nM and 1660 nM for EPHA2 and EPHA4, respectively.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Tyrosine Kinase
  • Target
    Ephrin Receptor
  • Recptor
    EPHA2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2245892-85-5
  • Formula Weight
    503.48
  • Molecular Formula
    C26H20F3N7O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:50 mg/mL (99.31 mM; Need ultrasonic);H2O:insoluble
  • SMILES
    O=C(NC1=CC=CC(C(F)(F)F)=C1)C2=CC=C(C)C(NC3=NC(C4=CC=CN=C4)=NC5=NN(C)C=C53)=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Tr?ster A, et al. NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family. ChemMedChem. 2018 Aug 20;13(16):1629-1633.
molnova catalog
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