GR 103691( —— )

Catalog No. M23720 CAS No. 162408-66-4

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	57	In Stock
2MG	33	In Stock
5MG	53	In Stock
10MG	93	In Stock
25MG	187	In Stock
50MG	299	In Stock
100MG	477	In Stock
200MG	677	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

GR 103691
Note

Research use only, not for human use.
Brief Description

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).
Description

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM). It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.
In Vitro

GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM).
In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Dopamine Receptor
Recptor

D3
Research Area

——
Indication

——

Chemical Information

CAS Number

162408-66-4
Formula Weight

485.62
Molecular Formula

C30H35N3O3
Purity

>98% (HPLC)
Solubility

DMSO:10 mM
SMILES

O=C(C1=CC=C(C2=CC=C(C(C)=O)C=C2)C=C1)NCCCCN3CCN(C4=CC=CC=C4OC)CC3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Audinot V, et al. A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J Pharmacol Exp Ther. 1998 Oct;287(1):187-97.

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