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Etripamil
CAS No. 1593673-23-4
Etripamil( MSP-2017 | (-)-MSP-2017 )
Catalog No. M23694 CAS No. 1593673-23-4
Etripamil displays atrioventricular nodal conduction and prolongs atrioventricular nodal refractory periods by inhibiting calcium ion influx through the calcium slow channels in the atrioventricular node cells. Etripamil is an antagonist of short-acting L-type calcium-channel.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 68 | In Stock |
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| 5MG | 112 | In Stock |
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| 10MG | 173 | In Stock |
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| 25MG | 312 | In Stock |
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| 50MG | 461 | In Stock |
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| 100MG | 693 | In Stock |
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| 200MG | 1088 | In Stock |
|
| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameEtripamil
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NoteResearch use only, not for human use.
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Brief DescriptionEtripamil displays atrioventricular nodal conduction and prolongs atrioventricular nodal refractory periods by inhibiting calcium ion influx through the calcium slow channels in the atrioventricular node cells. Etripamil is an antagonist of short-acting L-type calcium-channel.
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DescriptionEtripamil displays atrioventricular nodal conduction and prolongs atrioventricular nodal refractory periods by inhibiting calcium ion influx through the calcium slow channels in the atrioventricular node cells. Etripamil is an antagonist of short-acting L-type calcium-channel. It has a rapid onset of action designed for intranasal administration. It is also used to treat Paroxysmal Supraventricular Tachycardia.
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In Vitro——
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In Vivo——
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SynonymsMSP-2017 | (-)-MSP-2017
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorL-type calcium channel
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Research Area——
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Indication——
Chemical Information
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CAS Number1593673-23-4
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Formula Weight452.59
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Molecular FormulaC27H36N2O4
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Purity>98% (HPLC)
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SolubilityEthanol : 110 mg/mL (243.05 mM; Need ultrasonic)
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SMILESO=C(OC)C1=CC=CC(CCN(CCC[C@](C2=CC=C(OC)C(OC)=C2)(C#N)C(C)C)C)=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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L-Phenylalanine-15N
L-Phenylalanine-15N ((S)-2-Amino-3-phenylpropionic acid-15N) is the 15N-labeled L-Phenylalanine. L-Phenylalanine ((S)-2-Amino-3-phenylpropionic acid) is an essential amino acid isolated from Escherichia coli . L-Phenylalanine is a α2δ subunit of voltage-dependent Ca + channels antagonist with a K i of 980 nM.
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Cav 2.2 blocker 1
Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
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Mibefradil dihydroch...
Mibefradil dihydrochloride is an blocker of calcium channel with moderate selectivity for T-type Ca2+ channels (T-type and L-type currents with IC50s of 2.7 μM and 18.6 μM, respectively). Mibefradil dihydrochloride inhibits reversibly the T- and L-type currents with IC50 values of 2.7 and 18.6 μM, respectively.
