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Cav 2.2 blocker 1
CAS No. 1567335-29-8
Cav 2.2 blocker 1( —— )
Catalog No. M23678 CAS No. 1567335-29-8
Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 113 | In Stock |
|
| 5MG | 107 | In Stock |
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| 10MG | 183 | In Stock |
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| 25MG | 340 | In Stock |
|
| 50MG | 510 | In Stock |
|
| 100MG | 764 | In Stock |
|
| 200MG | 1004 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCav 2.2 blocker 1
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NoteResearch use only, not for human use.
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Brief DescriptionCav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
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DescriptionCav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorCav 2.2
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Research Area——
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Indication——
Chemical Information
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CAS Number1567335-29-8
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Formula Weight424.96
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Molecular FormulaC25H29ClN2O2
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Purity>98% (HPLC)
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SolubilityDMSO:20 mg/mL (47.07 mM; Need ultrasonic)
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SMILESCC1(C)CC(C2=NN(C3=CC=CC=C3OC)C(C4=CC=C(Cl)C=C4)=C2)CC(C)(C)O1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Wall MJ, et al. Discovery and optimization of a novel series of pyrazolyltetrahydropyran N-type calcium channel (Cav 2.2) blockers for the treatment of pain. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3780-3783.
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