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CYM 5520
CAS No. 1449747-00-5
CYM 5520( —— )
Catalog No. M23616 CAS No. 1449747-00-5
noncompetitive allosteric agonist of S1P2.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 100 | In Stock |
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| 2MG | 55 | In Stock |
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| 5MG | 90 | In Stock |
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| 10MG | 138 | In Stock |
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| 25MG | 250 | In Stock |
|
| 50MG | 365 | In Stock |
|
| 100MG | 546 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCYM 5520
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NoteResearch use only, not for human use.
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Brief Descriptionnoncompetitive allosteric agonist of S1P2.
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Descriptionnoncompetitive allosteric agonist of S1P2.
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In Vitro——
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In VivoAnimal Model:Ovariectomized 12 weeks old C57Bl6J mice Dosage:10 mg/kg.Administration:i.p.; 5 consecutive days per week; for 6 weeks Result:Corrected ovariectomy-induced osteopenia in mice by inducing new bone formation.
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Synonyms——
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PathwayGPCR/G Protein
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TargetS1P Receptor
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RecptorS1P2
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Research Area——
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Indication——
Chemical Information
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CAS Number1449747-00-5
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Formula Weight345.4
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Molecular FormulaC21H19N3O2
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Purity>98% (HPLC)
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SolubilityDMSO:≤30mg/ml
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SMILESCC1=CC(=C(N1CC2=CC=CC=C2)C)C(=O)CN3C=C(C=CC3=O)C#N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Satsu H , Schaeffer M T , Guerrero M , et al. A sphingosine 1-phosphate receptor 2 selective allosteric agonist[J]. Bioorganic & Medicinal Chemistry, 2013, 21( 17):5373-5382.
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