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SCD1 inhibitor-4
CAS No. 1295541-87-5
SCD1 inhibitor-4( —— )
Catalog No. M23453 CAS No. 1295541-87-5
SCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 65 | In Stock |
|
| 2MG | 36 | In Stock |
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| 5MG | 55 | In Stock |
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| 10MG | 101 | In Stock |
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| 25MG | 202 | In Stock |
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| 50MG | 319 | In Stock |
|
| 100MG | 458 | In Stock |
|
| 200MG | 637 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSCD1 inhibitor-4
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NoteResearch use only, not for human use.
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Brief DescriptionSCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.
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DescriptionSCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.
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In Vitro——
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In VivoSCD1 inhibitor-4 (1~30 mg/kg) shows a dose-dependent decrease in desaturation index with a 55 % reduction at 1 mg/kg and 85% reduction at the 10 and 30 mg/kg doses.
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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RecptorSCD1
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Research Area——
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Indication——
Chemical Information
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CAS Number1295541-87-5
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Formula Weight363.34
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Molecular FormulaC17H16F3N5O
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Purity>98% (HPLC)
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SolubilityDMSO: 90 mg/mL?(247.70 mM;?Need ultrasonic)
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SMILESO=C(C1=C(C)N(CC2=CC=CC(C(F)(F)F)=C2)C=N1)NC3=NN(C)C=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Atkinson KA, et al. N-benzylimidazole carboxamides as potent, orally active stearoylCoA desaturase-1 inhibitors. Bioorg Med Chem Lett. 2011;21(6):1621-1625.
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