BMS 182874 hydrochloride

CAS No. 1215703-04-0

BMS 182874 hydrochloride( —— )

Catalog No. M23383 CAS No. 1215703-04-0

BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 149 In Stock
2MG 93 In Stock
5MG 143 In Stock
10MG 216 In Stock
25MG 362 In Stock
50MG 494 In Stock
100MG 686 In Stock
200MG 926 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    BMS 182874 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.
  • Description
    BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Endothelin Receptor
  • Recptor
    ET-A
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1215703-04-0
  • Formula Weight
    381.88
  • Molecular Formula
    C17H20ClN3O3S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100mM
  • SMILES
    CC1=C(NS(=O)(C2=CC=CC3=C2C=CC=C3N(C)C)=O)ON=C1C.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.MARIA L WEBB, J. EILEEN BIRD, EDDIE C. K. LIU, PATRICIA M. ROSE, RANDY SERAFINO, PHILIP D. STEIN and SUZANNE MORELAND. BMS-182874 is a selective, nonpeptide endothelin ETA receptor antagonist. JPET 272:1124-1134, 1995.
molnova catalog
related products
  • Nebentan potassium

    Nebentan potassium (YM598) is an orally active and selective nonpeptide endothelin receptor (ETA receptor) antagonist.

  • Macitentan

    Macitentan is an orally active, non-peptide, dual ETA/ETB (endothelin) receptor antagonist with IC50 of 0.5 nM/391 nM.

  • Sitaxsentan sodium

    A potent, long acting, orally active, selective ETA receptor antagonist that binds competitively to human ETA receptor with Ki of 0.43 nM, IC50 of 1.4 nM.