MKC3946

CAS No. 1093119-54-0

MKC3946( —— )

Catalog No. M23297 CAS No. 1093119-54-0

MKC3946 is an effective and soluble IRE1α inhibitor which triggered modest growth inhibition in multiple myeloma cell lines.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 106 In Stock
2MG 64 In Stock
5MG 93 In Stock
10MG 155 In Stock
25MG 312 In Stock
50MG 461 In Stock
100MG 693 In Stock
200MG 918 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    MKC3946
  • Note
    Research use only, not for human use.
  • Brief Description
    MKC3946 is an effective and soluble IRE1α inhibitor which triggered modest growth inhibition in multiple myeloma cell lines.
  • Description
    MKC3946 is an effective and soluble IRE1α inhibitor which triggered modest growth inhibition in multiple myeloma cell lines.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    IRE1α
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1093119-54-0
  • Formula Weight
    380.46
  • Molecular Formula
    C21H20N2O3S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:30 mg/mL (78.85 mM)
  • SMILES
    CN1CCN(CC1)C(=O)C2=CC=C(S2)C3=CC4=C(C=C3)C(=C(C=C4)O)C=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Sun H, et al. Inhibition of IRE1α-driven pro-survival pathways is a promising therapeutic application in acute myeloid leukemia. Oncotarget. 2016 Apr 5;7(14):18736-49.
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