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PKC-iota inhibitor 1
CAS No. 2328094-11-5
PKC-iota inhibitor 1( —— )
Catalog No. M22982 CAS No. 2328094-11-5
PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 239 | In Stock |
|
| 2MG | 155 | In Stock |
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| 5MG | 231 | In Stock |
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| 10MG | 369 | In Stock |
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| 25MG | 616 | In Stock |
|
| 50MG | 861 | In Stock |
|
| 100MG | 1172 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 2344 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePKC-iota inhibitor 1
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NoteResearch use only, not for human use.
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Brief DescriptionPKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM).
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DescriptionPKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetPKC
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RecptorPKC-ι
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Research Area——
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Indication——
Chemical Information
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CAS Number2328094-11-5
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Formula Weight374.4
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Molecular FormulaC21H22N6O
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL?(333.83 mM;?Need ultrasonic)
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SMILESO=C(C1=CC(C2=CC=CC(N3CCNCC3)=C2)=CN=C1N)NC4=CC=NC=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kwiatkowski J, et al. Fragment-based Discovery of a Small-Molecule Protein Kinase C-iota Inhibitor Binding Post-kinase Domain Residues. ACS Med Chem Lett. 2019 Feb 15;10(3):318-323.
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