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Decoglurant (RO4995819)
CAS No. 911115-16-7
Decoglurant (RO4995819) ( RO4995819 )
Catalog No. M21765 CAS No. 911115-16-7
Decoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3. Decoglurant is developed as an antidepressant.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 147 | In Stock |
|
| 5MG | 222 | In Stock |
|
| 10MG | 357 | In Stock |
|
| 25MG | 597 | In Stock |
|
| 50MG | 851 | In Stock |
|
| 100MG | 1152 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDecoglurant (RO4995819)
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NoteResearch use only, not for human use.
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Brief DescriptionDecoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3. Decoglurant is developed as an antidepressant.
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DescriptionDecoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3. Decoglurant is developed as an antidepressant.
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In Vitro——
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In Vivo——
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SynonymsRO4995819
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PathwayGPCR/G Protein
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TargetmGluR
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number911115-16-7
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Formula Weight447.34
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Molecular FormulaC??H??F?N?
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Purity>98% (HPLC)
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SolubilityDMSO : 250 mg/mL (558.86 mM; Need ultrasonic)
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SMILESNC1=NC=C(C#CC2=C3N=C(C4=CC=C(C(F)(F)F)C=C4)C=C(C(F)(F)F)N3N=C2)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Wilkinson ST, et al. A new generation of antidepressants: an update on the pharmaceutical pipeline for novel and rapid-acting therapeutics in mood disorders based on glutamate/GABA neurotransmitter systems. Drug Discov Today. 2019 Feb;24(2):606-615.
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